The synthesis and SAR of novel diarylsulfone 11β-HSD1 inhibitors

Xuelei Yan; Zhong Lin Wang; Athena Sudom; Mario Cardozo; Michael DeGraffenreid; Yongmei Di; Pingchen Fan; Xiaodong He; Juan C. Jaén; Marc Labelle; Jinsong Liu; Ji Ma; Dustin L. McMinn; Shichang Miao; Daqing Sun; Liang Tang; Hua Tu; Stefania Ursu; Nigel P.C. Walker; Qiuping Ye; Jay P. Powers

doi:10.1016/j.bmcl.2010.09.097

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The synthesis and SAR of novel diarylsulfone 11β-HSD1 inhibitors

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