Synthesis and optimization of novel 4,4-disubstituted cyclohexylbenzamide derivatives as potent 11β-HSD1 inhibitors

Daqing Sun; Zhong Lin Wang; Seb Caille; Michael DeGraffenreid; Felix González-López de Turiso; Randall W. Hungate; Juan C. Jaén; Ben Jiang; Lisa D. Julian; Ron C. Kelly; Dustin L. McMinn; Jacob A. Kaizerman; Yosup Rew; Athena Sudom; Hua Tu; Stefania Ursu; Nigel P.C. Walker; Maren Gulsrud Willcockson; Xuelei Yan; Qiuping Ye; Jay P. Powers

doi:10.1016/j.bmcl.2010.10.129

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