Synthesis and optimization of arylsulfonylpiperazines as a novel class of inhibitors of 11β-hydroxysteroid dehydrogenase type 1 (11β-HSD1)

Daqing Sun; Zhong Lin Wang; Mario Cardozo; Rebekah Choi; Michael DeGraffenreid; Yongmei Di; Xiaodong He; Juan C. Jaén; Marc Labelle; Jinsong Liu; Ji Ma; Shichang Miao; Athena Sudom; Liang Tang; Hua Tu; Stefania Ursu; Nigel P.C. Walker; Xuelei Yan; Qiuping Ye; Jay P. Powers

doi:10.1016/j.bmcl.2008.12.114

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