Optimization of novel di-substituted cyclohexylbenzamide derivatives as potent 11β-HSD1 inhibitors

Dustin L. McMinn; Yosup Rew; Athena Sudom; Seb Caille; Michael DeGraffenreid; Xiaodong He; Randall W. Hungate; Ben Jiang; Juan C. Jaén; Lisa D. Julian; Jacob A. Kaizerman; Perry M. Novak; Daqing Sun; Hua Tu; Stefania Ursu; Nigel P.C. Walker; Xuelei Yan; Qiuping Ye; Zhong Lin Wang; Jay P. Powers

doi:10.1016/j.bmcl.2009.01.026

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