Discovery and Initial SAR of Arylsulfonylpiperazine Inhibitors of 11β-Hydroxysteroid Dehydrogenase Type 1 (11β-HSD1)

Daqing Sun; Zhong Lin Wang; Yongmei Di; Juan C. Jaén; Marc Labelle; Ji Ma; Shichang Miao; Athena Sudom; Liang Tang; Craig S. Tomooka; Hua Tu; Stefania Ursu; Nigel P.C. Walker; Xuelei Yan; Qiuping Ye; Jay P. Powers

doi:10.1016/j.bmcl.2008.05.025

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