Synthesis of New Homo and Heterodimers of 2′,3′-Dideoxyinosine (ddi) Using Ester Linkages

L. Ait Mohamed; Moha Taourirte; A. Rochdi; Hassan B. Lazrek; Jean‐Jacques Vasseur; J. W. Engels; Christophe Pannecouque; De Clercq Erik

doi:10.1081/ncn-120022664

Abstract

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A series of new homo and heterodimers of ddI has been synthesized. A glutarate diester spacer was used to covalently couple ddI onto ddI, AZT or d4T.

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