Exploiting the hydrophobic channel of the NNIBP: Discovery of novel diarylpyrimidines as HIV-1 NNRTIs against wild-type and K103N mutant viruses

Zhipeng Fu; Tao Zhang; Zhongxia Zhou; Dongwei Kang; Lin Sun; Shenghua Gao; Srinivasulu Cherukupalli; De Clercq Erik; Christophe Pannecouque; Xinyong Liu; Peng Zhan

doi:10.1016/j.bmc.2021.116239

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