Discovery of potent, selective, and orally bioavailable inhibitors of interleukin-1 receptor-associate kinase-4

Zhong Lin Wang; Daqing Sun; Sheree Johnstone; Zhaodan Cao; Xiong Gao; Juan C. Jaén; Jingqian Liu; Sarah Lively; Shichang Miao; Athena Sudom; Craig S. Tomooka; Nigel P.C. Walker; Matthew Wright; Xuelei Yan; Qiuping Ye; Jay P. Powers

doi:10.1016/j.bmcl.2015.10.060

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