Design, synthesis, and antiviral evaluation of novel piperidine-substituted arylpyrimidines as HIV-1 NNRTIs by exploring the hydrophobic channel of NNIBP

Tao Zhang; Zhongxia Zhou; Waleed A. Zalloum; Zhao Wang; Zhipeng Fu; Srinivasulu Cherukupalli; Da Feng; Yanying Sun; Shenghua Gao; De Clercq Erik; Christophe Pannecouque; Dongwei Kang; Peng Zhan; Xinyong Liu

doi:10.1016/j.bioorg.2021.105353

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De Clercq Erik

KU Leuven

Design, synthesis, and antiviral evaluation of novel piperidine-substituted arylpyrimidines as HIV-1 NNRTIs by exploring the hydrophobic channel of NNIBP

Article 2021 en

Authors

TZ
Tao Zhang
ZZ
Zhongxia Zhou
WZ
Waleed A. Zalloum

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Design, synthesis, and antiviral evaluation of novel piperidine-substituted arylpyrimidines as HIV-1 NNRTIs by exploring the hydrophobic channel of NNIBP

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