Unexpected Results in the Reaction of 5′-Tosyl TSAO-m<sup>3</sup>T With Amines

Clara Ibel Chamorro; Sonsoles Velázquez; M. Luísa Jimeno; María‐Jesús Pérez‐Pérez; Esther Lobatón; V. Tuñón; A. Esteban-gamboa; Federico Gago; De Clercq Erik; Jan Balzarini; Marı́a-José Camarasa; Ana San‐Félix

doi:10.1080/15257779908041551

Abstract

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Abstract We report our strategies to prepare TSAO compounds carrying at 5′-position groups, such as amines, that may be positively charged at physiological conditions, unexpectedly, cyclic TSAO-derivatives were obtained. A possible mechanism for the formation of these unexpected compounds is advanced.

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