Towards new C6-rigid S-DABO HIV-1 reverse transcriptase inhibitors: Synthesis, biological investigation and molecular modeling studies

Hai-Qiu Wu; Zihong Yan; Wenxue Chen; Qiuqin He; Fen‐Er Chen; De Clercq Erik; Jan Balzarini; Dirk Daelemans; Christophe Pannecouque

doi:10.1016/j.bmc.2013.08.040

Back

Towards new C6-rigid S-DABO HIV-1 reverse transcriptase inhibitors: Synthesis, biological investigation and molecular modeling studies

Article 2013 en

Discussion(0)

No comments yet. Be the first to comment.

Related publications

Article2014

Synthesis and biological evaluation of new conformationally restricted S-DABO hybrids as non-nucleoside inhibitors of HIV-1 reverse transcriptase

Hai-Qiu Wu, Christophe Pannecouque, Zihong Yan, Wenxue Chen, Qiuqin He, Fen‐Er Chen, Jan Balzarini, Dirk Daelemans, De Clercq Erik

Article2023

Design, synthesis, and biological testing of biphenylmethyloxazole inhibitors targeting HIV-1 reverse transcriptase

Zachary J. Carter, Klarissa Hollander, Krasimir A. Spasov, Karen S. Anderson, William L. Jorgensen

Bioorganic & Medicinal Chemistry Letters

Article2014

Synthesis and biological evaluation of CHX-DAPYs as HIV-1 non-nucleoside reverse transcriptase inhibitors

Zihong Yan, Hai-Qiu Wu, Wenxue Chen, Yan Wu, Hu‐Ri Piao, Qiuqin He, Fen‐Er Chen, De Clercq Erik, Christophe Pannecouque

Article1992

Specific HIV-1 Reverse Transcriptase Inhibitors

Zeger Debyser, Rudi Pauwels, Koen Andries, De Clercq Erik

Article2001

Synthesis, Biological Activity, Pharmacokinetic Properties and Molecular Modelling Studies of Novel 1H,3H-Oxazolo[3,4-a]Benzimidazoles: Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitors

Alba Chimirri, Pierre Monforte, Angela Rao, Maria Zappalà, AM Monforte, Giovambattista De Sarro, Christophe Pannecouque, Myriam Witvrouw, Jan Balzarini, De Clercq Erik