Synthesis of Acycloalkenyl Derivatives of Pyrimidines and Purines

Hassan B. Lazrek; N. Redwane; A. Rochdi; J. L. Barascut; J.‐L. IMBACH; De Clercq Erik

doi:10.1080/15257779508012380

Abstract

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Abstract Conjugate addition of an anionic nucleophile (nucleobase) to an active triple bond (α, β unsaturated carboxylate or phosphonate) was used for preparing α-ethenyl carboxylate or phosphonate derivatives of purines and pyrimidines.

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