Synthesis and Anti-HIV Activity of Dideoxycytidine Analogues Containing a Pyranose Carbohydrate Moiety

Arthur Van Aerschot; L. Kerremans; Jan Balzarini; De Clercq Erik; Piet Herdewijn

doi:10.1080/07328319108046539

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Synthesis and Anti-HIV Activity of Dideoxycytidine Analogues Containing a Pyranose Carbohydrate Moiety

Article 1991 en

Abstract

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Abstract Dideoxycytidine analogues with a trideoxy-D-hexopyranosyl or hexenopyranosyl moiety were synthesized starting from 2-deoxyglucosyl bromide or tri-O-acetyl-D-glucal.

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