Inhibiting NF-κB-inducing kinase (NIK): Discovery, structure-based design, synthesis, structure–activity relationship, and co-crystal structures

Kexue Li; Lawrence R. McGee; Ben Fisher; Athena Sudom; Jun S. Liu; Steven M. Rubenstein; Mohmed K. Anwer; Timothy D. Cushing; Youngsook Shin; Merrill Ayres; Fei Lee; John Eksterowicz; Paul Faulder; Bohdan Waszkowycz; Olga Plotnikova; Ellyn Farrelly; Shou-Hua Xiao; Guoqing Chen; Zhong Lin Wang

doi:10.1016/j.bmcl.2013.01.012

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Inhibiting NF-κB-inducing kinase (NIK): Discovery, structure-based design, synthesis, structure–activity relationship, and co-crystal structures

Article 2013 en

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Inhibiting NF-κB-inducing kinase (NIK): Discovery, structure-based design, synthesis, structure–activity relationship, and co-crystal structures

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