Identification and optimization of N3,N6-diaryl-1H-pyrazolo[3,4-d]pyrimidine-3,6-diamines as a novel class of ACK1 inhibitors

David J. Kopecky; Xiaolin Hao; Yi Chen; Jiasheng Fu; Xian‐Yun Jiao; Juan C. Jaén; Mario Cardozo; Jinsong Liu; Zhong Lin Wang; Nigel P.C. Walker; Holger Wesche; Shyun Li; Ellyn Farrelly; Shou-Hua Xiao; Frank Kayser

doi:10.1016/j.bmcl.2008.10.092

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Identification and optimization of N3,N6-diaryl-1H-pyrazolo[3,4-d]pyrimidine-3,6-diamines as a novel class of ACK1 inhibitors

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