Discovery of novel piperidine-substituted indolylarylsulfones as potent HIV NNRTIs via structure-guided scaffold morphing and fragment rearrangement

Xiao Li; Ping Gao; Boshi Huang; Zhongxia Zhou; Yu Zhao; Yuan Zheng; Huiqing Liu; Christophe Pannecouque; Dirk Daelemans; De Clercq Erik; Peng Zhan; Xinyong Liu

doi:10.1016/j.ejmech.2016.10.009

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Discovery of novel piperidine-substituted indolylarylsulfones as potent HIV NNRTIs via structure-guided scaffold morphing and fragment rearrangement

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