Discovery of novel diarypyrimidine derivatives as potent HIV-1 NNRTIs by exploiting the tolerant region I within NNRTI binding pocket

Xiangkai Ji; Xiangyi Jiang; Zhen Gao; Heng Gao; De Clercq Erik; Christophe Pannecouque; Dongwei Kang; Shujing Xu; Xinyong Liu

doi:10.1016/j.ejmech.2025.117787

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