Design, synthesis and evaluation of novel HIV-1 NNRTIs with dual structural conformations targeting the entrance channel of the NNRTI binding pocket

Qing Meng; Xuwang Chen; Dongwei Kang; Boshi Huang; Wenxin Li; Peng Zhan; Dirk Daelemans; De Clercq Erik; Christophe Pannecouque; Xinyong Liu

doi:10.1016/j.ejmech.2016.02.068

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Design, synthesis and evaluation of novel HIV-1 NNRTIs with dual structural conformations targeting the entrance channel of the NNRTI binding pocket

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Design, synthesis and evaluation of novel HIV-1 NNRTIs with dual structural conformations targeting the entrance channel of the NNRTI binding pocket

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