Design, synthesis and bioevaluation of novel maleamic amino acid ester conjugates of 3,5-bisarylmethylene-4-piperidones as cytostatic agents

Dani Youssef; Elizabeth Potter; Mamta Jha; De Clercq Erik; Jan Balzarini; James P. Stables; Amitabh Jha

doi:10.1016/j.bmcl.2009.09.069

Related publications

Article2003

3,5-Bis(Phenylmethylene)-1-(N-arylmaleamoyl)-4-piperidones: A Novel Group of Cytotoxic Agents

Jonathan R. Dimmock, Amitabh Jha, Gordon A. Zello, Rajendra K. Sharma, Anuraag Shrivastav, Selvakumar Palaniappan, Theresa M. Allen, C.L. Santos, Jan Balzarini, De Clercq Erik, Elias K. Manavathu, James P. Stables

Article2006

Design, synthesis and cytotoxic properties of novel 1-[4-(2-alkylaminoethoxy)phenylcarbonyl]-3,5-bis(arylidene)-4-piperidones and related compounds

Umashankar Das, Jane Alcorn, Anuraag Shrivastav, Rajendra K. Sharma, De Clercq Erik, Jan Balzarini, Jonathan R. Dimmock

Article2016

3,5-Bis(3-alkylaminomethyl-4-hydroxybenzylidene)-4-piperidones: A Novel Class of Potent Tumor-Selective Cytotoxins

Subhas S. Karki, Umashankar Das, Naoki Umemura, Hiroshi Sakagami, Shoko Iwamoto, Masami Kawase, Jan Balzarini, De Clercq Erik, Stephen G. Dimmock, Jonathan R. Dimmock

Article2014

Microwave assisted synthesis and QSAR study of novel NSAID acetaminophen conjugates with amino acid linkers

Anand D. Tiwari, Siva S. Panda, Adel S. Girgis, Sandhyamayee Sahu, Riham F. George, Aladdin M. Srour, Brian La Starza, Abdullah Mohamed Asiri, C. Dennis Hall, Alan R. Katritzky

Article1998

Retinoids as potential chemotherapeutic agents. Synthesis, cytostatic and differentiating activities of new heterocyclic analogs of retinoic acid

Stefano Manfredini, Daniele Simoni, Giuseppe Caminiti, Silvia Vertuani, Francesco Paolo Invidiata, L Moscato, Sigrid Hatse, De Clercq Erik, Jan Balzarini