1-Hydroxypyrido[2,3-d]pyrimidin-2(1H)-ones as novel selective HIV integrase inhibitors obtained via privileged substructure-based compound libraries

Ping Gao; Lingzi Zhang; Lin Sun; Tianguang Huang; Jing Tan; Jian Zhang; Zhongxia Zhou; Tong Zhao; Luis Menéndez‐Arias; Christophe Pannecouque; De Clercq Erik; Peng Zhan; Xinyong Liu

doi:10.1016/j.bmc.2017.09.006

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1-Hydroxypyrido[2,3-d]pyrimidin-2(1H)-ones as novel selective HIV integrase inhibitors obtained via privileged substructure-based compound libraries

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